中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
机构
  • 上海药物研究所 [10]
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内容类型
发表日期
  • 2022 [10]
学科主题
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浏览/检索结果: 共10条,第1-10条 帮助

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Structure-Based Design of Tropane Derivatives as a Novel Series of CCR5 Antagonists with Broad-Spectrum Anti-HIV-1 Activities and Improved Oral Bioavailability 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 24, 页码: 16526-16540
作者:  
Xie, Xiong;  Zheng, Yu-Gui;  Chen, Huan;  Li, Jian;  Luo, Rong-Hua
  |  收藏  |  浏览/下载:26/0  |  提交时间:2023/04/10
Loss of VOPP1 Contributes to BET Inhibitor Acquired Resistance in Non-Small Cell Lung Cancer Cells 期刊论文  OAI收割
MOLECULAR CANCER RESEARCH, 2022, 卷号: 20, 期号: 12, 页码: 1785-1798
作者:  
Sun, Lin;  Wu, Qian;  Huan, Xia-Juan;  Tian, Chang-Qing;  Wang, Ying-Qing
  |  收藏  |  浏览/下载:14/0  |  提交时间:2024/03/21
SOMCL-19-133, a novel, selective, and orally available inhibitor of NEDD8-activating enzyme (NAE) for cancer therapy 期刊论文  OAI收割
NEOPLASIA, 2022, 卷号: 32, 页码: 12
作者:  
Zhou, Li-Na;  Xiong, Chaodong;  Cheng, Yong-Jun;  Song, Shan-Shan;  Bao, Xu-Bin
  |  收藏  |  浏览/下载:14/0  |  提交时间:2023/04/10
Design and development of a novel series of oral bivalent BET inhibitors with potent anticancer activities 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 239, 页码: 13
作者:  
Luo, Menglan;  Wu, Qian;  Yang, Yueyue;  Sun, Lin;  Huan, Xiajuan
  |  收藏  |  浏览/下载:40/0  |  提交时间:2022/08/30
Pharmacokinetics, mass balance, and metabolism of [C-14]TPN171, a novel PDE5 inhibitor, in humans for the treatment of pulmonary arterial hypertension 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2022, 页码: 13
作者:  
He, Yi-fei;  Liu, Yin;  Yu, Jing-hua;  Cheng, Huan;  Odilov, Abdullajon
  |  收藏  |  浏览/下载:31/0  |  提交时间:2022/08/16

Design, synthesis, and biological evaluations of substituted pyrazoles as pyrrolomycin analogues against staphylococcal biofilm & nbsp;

期刊论文  OAI收割

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 236, 页码: 13
作者:  
Huan, Xiang;  Wang, Yanhui;  Peng, Xiaofeng;  Xie, Shanshan;  He, Qian
  |  收藏  |  浏览/下载:30/0  |  提交时间:2022/08/16
New laboratory evidence for the association between endothelial dysfunction and COVID-19 disease progression 期刊论文  OAI收割
JOURNAL OF MEDICAL VIROLOGY, 2022, 页码: 9
作者:  
Liu, Nan;  Long, Hui;  Sun, Jianhua;  Li, Huan;  He, Yunting
  |  收藏  |  浏览/下载:25/0  |  提交时间:2022/06/15
The novel therapeutic strategy of vilazodone-donepezil chimeras as potent triple-target ligands for the potential treatment of Alzheimer's disease with comorbid depression 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 229, 页码: 22
作者:  
Li, Xiaokang;  Li, Jinwen;  Huang, Yunyuan;  Gong, Qi;  Fu, Yan
  |  收藏  |  浏览/下载:32/0  |  提交时间:2022/06/15
Absorption, distribution, metabolism, and excretion of [C-14]TPN729 after oral administration to rats 期刊论文  OAI收割
XENOBIOTICA, 2022, 页码: 12
作者:  
Cheng, Huan;  Yu, Jinghua;  Yang, Chen;  Zhang, Ning;  Fan, Zhen
  |  收藏  |  浏览/下载:31/0  |  提交时间:2022/06/15
Metal-drug nanoparticles-mediated osteolytic microenvironment regulation for enhanced radiotherapy of orthotopic osteosarcoma (vol 417, 128103, 2021) 期刊论文  OAI收割
CHEMICAL ENGINEERING JOURNAL, 2022, 卷号: 428, 页码: 2
作者:  
Geng, Huan;  Zhou, Mengxue;  Li, Bin;  Liu, Liang;  Yang, Xu
  |  收藏  |  浏览/下载:35/0  |  提交时间:2022/01/18