中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共379条,第1-10条 帮助

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The Tyrosine Kinase Inhibitor Bafetinib Inhibits PAR2-induced Activation of TRPV4 In Vitro and Pain In Vivo1 期刊论文  OAI收割
出版物, 2111, 页码: 1-44
作者:  
1M S Grace;  T Lieu;  B Darby;  F C Abogadie;  N Veldhuis N W Bunnett;  P McIntyre
  |  收藏  |  浏览/下载:226/0  |  提交时间:2017/07/24
Discovery of a Covalent Inhibitor Selectively Targeting the Autophosphorylation Site of c-Src Kinase 期刊论文  OAI收割
ACS CHEMICAL BIOLOGY, 2024, 页码: 12
作者:  
Zhang, Huimin;  Xu, Dounan;  Huang, Hongchan;  Jiang, Hao;  Hu, Linghao
  |  收藏  |  浏览/下载:1/0  |  提交时间:2024/05/07
Pharmacokinetics, mass balance, and metabolism of [14C]envonalkib (TQ-B3139), a novel ALK tyrosine kinase inhibitor, in healthy Chinese subjects 期刊论文  OAI收割
CANCER CHEMOTHERAPY AND PHARMACOLOGY, 2024, 页码: 11
作者:  
Ma, Sheng;  Wang, Xin;  Yan, Shu;  Miao, Liyan;  Wan, Xiaojing
  |  收藏  |  浏览/下载:4/0  |  提交时间:2024/05/07
Discovery of a 1,6-naphthyridin-4-one-based AXL inhibitor with improved pharmacokinetics and enhanced in vivo antitumor efficacy 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 265, 页码: 17
作者:  
Lan, Yaohan;  Peng, Xia;  Ji, Yinchun;  Su, Yi;  Duan, Wenhu
  |  收藏  |  浏览/下载:12/0  |  提交时间:2024/02/27
Discovery of a potent and selective covalent threonine tyrosine kinase (TTK) inhibitor 期刊论文  OAI收割
BIOORGANIC CHEMISTRY, 2024, 卷号: 143, 页码: 16
作者:  
Sun, Yaoliang;  Chen, Zhiwen;  Liu, Guobin;  Chen, Xiaoai;  Shi, Zihan
  |  收藏  |  浏览/下载:13/0  |  提交时间:2024/03/25
KinomeMETA: meta-learning enhanced kinome-wide polypharmacology profiling 期刊论文  OAI收割
BRIEFINGS IN BIOINFORMATICS, 2024, 卷号: 25, 期号: 1, 页码: 15
作者:  
Ren, Qun;  Qu, Ning;  Sun, Jingjing;  Zhou, Jingyi;  Liu, Jin
  |  收藏  |  浏览/下载:1/0  |  提交时间:2024/05/07
Structure-based drug discovery of novel fused- pyrazolone carboxamide derivatives as potent and selective AXL inhibitors 期刊论文  OAI收割
ACTA PHARMACEUTICA SINICA B, 2023, 卷号: 13, 期号: 12, 页码: 4918-4933
作者:  
Fang, Feifei;  Dai, Yang;  Wang, Hao;  Ji, Yinchun;  Liang, Xuewu
  |  收藏  |  浏览/下载:8/0  |  提交时间:2024/01/26
Design, synthesis and pharmacological evaluation of 2,3-dihydrobenzo-furan IRAK4 inhibitors for the treatment of diffuse large B-cell lymphoma 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 256, 页码: 16
作者:  
Chen, Yun;  Ning, Yi;  Chen, Zhiwei;  Xue, Yaping;  Wu, Qingyun
  |  收藏  |  浏览/下载:12/0  |  提交时间:2023/10/17
Pharmaco-proteogenomic characterization of liver cancer organoids for precision oncology 期刊论文  OAI收割
SCIENCE TRANSLATIONAL MEDICINE, 2023, 卷号: 15, 期号: 706, 页码: 15
作者:  
Ji, Shuyi;  Feng, Li;  Fu, Zile;  Wu, Gaohua;  Wu, Yingcheng
  |  收藏  |  浏览/下载:15/0  |  提交时间:2023/10/17
Traditional Chinese Medicine Targeting Sarcoma Virus Oncogene-related Diseases 期刊论文  OAI收割
CURRENT CANCER DRUG TARGETS, 2023, 卷号: 23, 期号: 10, 页码: 751-763
作者:  
Wang, Yiying;  Wang, Xiaoyu;  Su, Kexin;  Yang, Yifu
  |  收藏  |  浏览/下载:9/0  |  提交时间:2023/10/17