机构

• 上海药物研究所 [5]
• 化学研究所 [2]
• 中国科学院大学 [1]

采集方式

• OAI收割 [7]
• iSwitch采集 [1]

内容类型

• 期刊论文 [8]

发表日期

• 2022 [1]
• 2021 [2]
• 2014 [1]
• 2010 [1]
• 2008 [1]
• 2006 [1]
• 更多

学科主题

筛选

浏览/检索结果: 共8条，第1-8条 帮助 条数/页： 5101520253035404550556065707580859095100 排序方式： 请选择题名升序题名降序提交时间升序提交时间降序作者升序作者降序发表日期升序发表日期降序 Identification of 1H-pyrazolo[3,4-b]pyridine derivatives as novel and potent TBK1 inhibitors: design, synthesis, biological evaluation, and molecular docking study 期刊论文  OAI收割 JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 2022, 卷号: 37, 期号: 1, 页码: 1411-1425 作者:  Sun, Yin;  Tang, Haotian;  Wang, Xiaoyan;  Feng, Fang;  Fan, Tiantian   |  收藏  |  浏览/下载：55/0  |  提交时间：2022/08/16 TBK1 inhibitors  1H-pyrazolo[3  4-b]pyridine  structure-activity relationships (SARs)  immune response  cancer therapy   Discovery and structure - activity relationship exploration of pyrazolo [1,5-a]pyrimidine derivatives as potent FLT3-ITD inhibitors 期刊论文  OAI收割 BIOORGANIC & MEDICINAL CHEMISTRY, 2021, 卷号: 48, 页码: 13 作者:  Chen, Yun;  Bai, Gang;  Li, Yan;  Ning, Yi;  Cao, Sufen   |  收藏  |  浏览/下载：70/0  |  提交时间：2021/12/01 FLT3  FLT3-ITD  Acute myeloid leukemia  Structure-activity relationships  Pyrazolo[1, 5-a]pyrimidine   Synthesis and Evaluation of 3-(Indol-3-yl)-4-(Pyrazolo[3,4-c]Pyridazin-3-yl)-Maleimides as Potent Mutant Isocitrate Dehydrogenase-1 Inhibitors 期刊论文  OAI收割 PHARMACEUTICAL CHEMISTRY JOURNAL, 2021, 卷号: 55, 期号: 7, 页码: 655-664 作者:  Xu, Jianghong;  Hu, Yuanyuan;  Liu, Xiaoqi;  Gao, Anhui;  Gao, Lixin   |  收藏  |  浏览/下载：55/0  |  提交时间：2021/12/01 IDH1-R132H inhibitors  synthesis  biological activity  docking  3-(indol-3-yl)-4-(pyrazolo-[3  4-c]pyridazin-3-yl)-maleimides   Synthesis of Pyrazolo[1,2-a] cinnolines via a Rhodium-Catalyzed Oxidative Coupling Approach 期刊论文  OAI收割 ADVANCED SYNTHESIS & CATALYSIS, 2014, 卷号: 356, 期号: 5, 页码: 972-976 作者:  Xing, Li;  Fan, Zhoulong;  Hou, Chengyu;  Yong, Guoping;  Zhang, Ao   |  收藏  |  浏览/下载：20/0  |  提交时间：2019/01/08 alkynes  oxidative coupling  pyrazolo[1  2-a]cinnolines  pyrazolones  rhodium   Design and synthesis of 1,4,5,6-tetrahydropyrrolo[3,4-c]pyrazoles and pyrazolo[3,4-b]pyridines for Aurora-A kinase inhibitors 期刊论文  OAI收割 BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2010, 卷号: 20, 期号: 14, 页码: 4273-4278 作者:  Shi, Jianyou;  Xu, Guobin;  Zhu, Wei;  Ye, Haoyu;  Yang, Shengyong   |  收藏  |  浏览/下载：38/0  |  提交时间：2019/01/08 1,4,5,6-Tetrahydropyrrolo[3,4-c]pyrazoles  Pyrazolo[3,4-b]pyridines  Antitumor  Aurora-A kinase   Efficient construction of pyrazolo[1,5-a]pyrimidine scaffold and its exploration as a new heterocyclic fluorescent platform 期刊论文  OAI收割 JOURNAL OF FLUORESCENCE, 2008, 卷号: 18, 期号: 2, 页码: 357-363 作者:  Wu, Yan-Chao;  Li, Hui-Jing;  Liu, Li;  Wang, Dong;  Yang, Hua-Zheng   |  收藏  |  浏览/下载：25/0  |  提交时间：2019/04/09 Fluorophore  Heterocycle  Fluorescence  Pyrazolo[1  5-a]Pyrimidine   Synthesis of trifluoromethyl-promoted functional pyrazolo [1,5-a]pyrimidine and pyrazolo [5,1-d] [1,2,3,5]tetrazine-4(3H)-ones 期刊论文  OAI收割 JOURNAL OF FLUORINE CHEMISTRY, 2006, 卷号: 127, 期号: 3, 页码: 409-416 作者:  Wu, YC;  Chen, YJ;  Li, HJ;  Zou, XM;  Hu, FZ   |  收藏  |  浏览/下载：15/0  |  提交时间：2019/04/09 Fluorine  Pyrazole  Inhibitor  Pyrazolo[1  Pyrazolo[5  5-a]Pyrimidine  1-d][1  2  3  5]Tetrazine-4(3h)-one   Synthesis of 3-amino-6/8-substituted-1h-pyrazolo[4,3-c]quinolines 期刊论文  iSwitch采集 Chemical journal of chinese universities-chinese, 2005, 卷号: 26, 期号: 2, 页码: 250-253 作者:  Qiao, RZ;  Zhang, ZY;  Zhao, YF 收藏  |  浏览/下载：29/0  |  提交时间：2019/05/10 1,2,4-triazolo[3,4-b]-1,3,4-thiadiazole  3-amino-6/8-substituted-1h-pyrazolo[4,3-c] quinoline  Synthesis  Property