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Pharmacological characterizationof tachykinin tetrabranched derivatives
期刊论文
OAI收割
出版物, 3111, 期号: 0, 页码: 1-36
作者:
Chiara Ruzza
;
Anna Rizzi
;
Davide Malfacini
;
Maria Camilla Cerlesi
;
Federica Ferrari
  |  
收藏
  |  
浏览/下载:177/0
  |  
提交时间:2017/07/24
Tachykinins
Substance p
Pwt2-sp
Nk1 Receptor
Calcium Mobilization
Bioluminescence Resonance Energy Transfer
Guinea Pig Ileum
Rat Urinary Bladder
Nociceptive Behaviour Induced By Spinal Substance p
Mice
Rational design and discovery of novel oxalate-like derivatives as aphid-repellent candidates based on odorant-binding protein 3
期刊论文
OAI收割
JOURNAL OF MOLECULAR STRUCTURE, 2024, 卷号: 1301, 页码: 11
作者:
Zhu, Ziwei
;
Li, Jianing
;
Liu, Chong
;
Li, Huilin
;
Lu, Xingxing
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2024/04/09
Odorant-binding protein
Oxalate-like derivatives
Rational design
Repellent activity
Behavioural control agents
Discovery of betulinic acid derivatives as gut-restricted TGR5 agonists: Balancing the potency and physicochemical properties
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2024, 卷号: 144, 页码: 18
作者:
Zhuo, Ning
;
Yun, Ying
;
Zhang, Chenlu
;
Guo, Shimeng
;
Yin, Jianpeng
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2024/03/25
Type 2 Diabetes
TGR5 agonist
Betulinic acid
Gut-restricted
Gallbladder-filling effects
Kinetophores
Synthesis of 1,4-epoxy-2-aryltetrahydro-1-benzazepines
via
rhodium(
iii
)-catalyzed C-H allylation/intramolecular 1,3-dipolar cycloaddition
期刊论文
OAI收割
CHEMICAL COMMUNICATIONS, 2024, 卷号: 60, 期号: 17, 页码: 2401-2404
作者:
Wang, Xuan
;
Li, Jianlong
;
Du, Haifang
;
Liang, Weihong
;
Luo, Cheng
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2024/03/13
Synthesis and Characterization of Slow-Release Chitosan Oligosaccharide Pyridine Schiff Base Copper Complexes with Antifungal Activity
期刊论文
OAI收割
JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY, 2024, 卷号: 72, 期号: 8, 页码: 3872-3883
作者:
Liu, Weixiang
;
Qin, Yukun
;
Liu, Song
;
Xing, Ronge
;
Yu, Huahua
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2024/04/07
antifungal
chitosan oligosaccharide
coppercomplex
Schiff base
slow-release
Effective correction of dissolved organic carbon interference in nitrate detection using ultraviolet spectroscopy combined with the equivalent concentration offset method
期刊论文
OAI收割
RSC ADVANCES, 2024, 卷号: 14, 期号: 8, 页码: 5370-5379
作者:
Dong, Jing
;
Tang, Junwu
;
Wu, Guojun
;
Xin, Yu
;
Li, Ruizhuo
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2024/03/15
DRAK2 suppresses autophagy by phosphorylating ULK1 at Ser
56
to diminish pancreatic β cell function upon overnutrition
期刊论文
OAI收割
SCIENCE TRANSLATIONAL MEDICINE, 2024, 卷号: 16, 期号: 733, 页码: 16
作者:
Lu, Yuting
;
Xu, Junyu
;
Li, Yufeng
;
Wang, Ruoran
;
Dai, Chengqiu
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2024/03/13
Discovery of a brain-permeable bromodomain and extra terminal domain (BET) inhibitor with selectivity for BD1 for the treatment of multiple sclerosis
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 265, 页码: 14
作者:
Chen, Xuetao
;
Wu, Tingting
;
Du, Zhiyan
;
Kang, Wenjing
;
Xu, Rujun
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2024/02/27
BET
BD1
Bromodomain
Brain-permeable
Multiple sclerosis
Novel imidazo[1,2,4] triazole derivatives: Synthesis, fluorescence, bioactivity for SHP1
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 265, 页码: 15
作者:
Yan, Xue
;
Zhang, Chun
;
Gao, Li-Xin
;
Liu, Min -Min
;
Yang, Yu-Ting
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2024/02/27
Imidazo[124] triazole derivatives
Fluorescence property
SHP1
Bioactivity
Cellular imaging
Discovery of a 1,6-naphthyridin-4-one-based AXL inhibitor with improved pharmacokinetics and enhanced in vivo antitumor efficacy
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 265, 页码: 17
作者:
Lan, Yaohan
;
Peng, Xia
;
Ji, Yinchun
;
Su, Yi
;
Duan, Wenhu
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2024/02/27
AXL inhibitor
In vivo antitumor efficacy
6-Naphthyridin-4-one derivatives
Scaffold hopping
Structure-based drug design