中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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植物研究所 [18]
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Structure-based identification of new orally bioavailable BRD9-PROTACs for treating acute myelocytic leukemia
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 262, 页码: 18
作者:
Zhang, Jingyu
;
Duan, Haiting
;
Gui, Renzhao
;
Wu, Mingfei
;
Shen, Liteng
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2023/12/19
Acute myeloid leukemia
Bromodomain-containing protein 9
Proteolysis-targeting chimera
Orally bioavailable
Docking
Transcriptional regulation analysis reveals the complexity of metamorphosis in the Pacific oyster (Crassostrea gigas)
期刊论文
OAI收割
MARINE LIFE SCIENCE & TECHNOLOGY, 2023, 页码: 11
作者:
Xu, Fei
;
Deng, Shaoxi
;
Gavriouchkina, Daria
;
Zhang, Guofan
  |  
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2024/04/07
Gene regulation network
Indirect development
Lophotrochozoa
Nuclear receptors
Neurohormones
Protein synthesis
Transcription factors
Glutamine Production by Glul Promotes Thermogenic Adipocyte Differentiation Through Prdm9-Mediated H3K4me3 and Transcriptional Reprogramming
期刊论文
OAI收割
DIABETES, 2023, 卷号: 72, 期号: 11, 页码: 24
作者:
Pan, Xiaowen
;
Ye, Lingxia
;
Guo, Xiaozhen
;
Wang, Weihua
;
Zhang, Ziyin
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2024/03/25
Smilagenin induces expression and epigenetic remodeling of BDNF in alzheimer's disease
期刊论文
OAI收割
PHYTOMEDICINE, 2023, 卷号: 118, 页码: 11
作者:
Yang, Shuangshuang
;
Fan, Lei
;
Zhang, Rui
;
Song, Chenghuan
;
Shi, Jiyun
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2023/10/17
Alzheimer's disease
Brain-derived neurotrophic factor
Histone acetylation
Smilagenin
Discovery of new small molecule inhibitors of the BPTF bromodomain
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2023, 卷号: 134, 页码: 106453
作者:
Liang, Xiaochen
;
Cao, Yu
;
Duan, Zhe
;
Wang, Mingchen
;
Zhang, Naixia
  |  
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2024/03/27
BPTF bromodomain
BPTF inhibitors
HTRF
c-Myc
ARID1A loss induces polymorphonuclear myeloid-derived suppressor cell chemotaxis and promotes prostate cancer progression
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2022, 卷号: 13, 期号: 1, 页码: 20
作者:
Li, Ni
;
Liu, Qiuli
;
Han, Ying
;
Pei, Siyu
;
Cheng, Bisheng
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2023/04/10
HBO1 catalyzes lysine benzoylation in mammalian cells
期刊论文
OAI收割
ISCIENCE, 2022, 卷号: 25, 期号: 11, 页码: 14
作者:
Tan, Doudou
;
Wei, Wei
;
Han, Zhen
;
Ren, Xuelian
;
Yan, Cong
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2023/04/10
Vanguard is a Glucose Deprivation-Responsive Long Non-Coding RNA Essential for Chromatin Remodeling-Reliant DNA Repair
期刊论文
OAI收割
ADVANCED SCIENCE, 2022
作者:
Zhang, Ben
;
Thorne, Rick Francis
;
Zhang, Pengfei
;
Wu, Mian
;
Liu, Lianxin
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2022/12/23
genomic stability
HMGB1
long non-coding RNAs
PARP inhibitors
Vanguard
Discovery of a highly potent CECR2 bromodomain inhibitor with 7H-pyrrolo[2,3-d] pyrimidine scaffold
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2022, 卷号: 123, 页码: 12
作者:
Lu, Haibo
;
Lu, Tian
;
Zu, Shijia
;
Duan, Zhe
;
Guang, Yiman
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2022/08/16
CECR2 bromodomain
BPTF bromodomain
Small-molecule inhibitor
SAR study
Chemical probe
Histone acetyltransferase GCN5-mediated lysine acetylation modulates salt stress aadaption of Trichoderma
期刊论文
OAI收割
APPLIED MICROBIOLOGY AND BIOTECHNOLOGY, 2022, 卷号: 106, 期号: 8, 页码: 3033-3049
作者:
Li, Zhe
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2022/11/08
NUCLEOTIDE EXCISION-REPAIR
PROGRAMMED CELL-DEATH
MEMBRANE H+-ATPASE
OXIDATIVE STRESS
GROWTH
GCN5
TRANSPORT
SALINITY
REESEI
METABOLISM