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Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [40]
采集方式
OAI收割 [40]
内容类型
期刊论文 [38]
会议论文 [2]
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2023 [3]
2022 [2]
2021 [1]
2020 [2]
2019 [3]
2018 [2]
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专题:上海药物研究所
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Discovery of zolinium TSG1180 as a novel agonist of transgelin-2 for treating asthma
期刊论文
OAI收割
Biomedicine & pharmacotherapy = Biomedecine & pharmacotherapie, 2023, 卷号: 167, 页码: 115556
作者:
Yuan, Hong-Kai
;
Li, Bo
;
Wu, Leyun
;
Wang, Xue-Ling
;
Lv, Zhi-Ying
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2024/03/26
Active learning
Consensus labelling
Eye irritation
Serious eye damage
Structural alerts
AXL antibody and AXL-ADC mediate antitumor efficacy via targeting AXL in tumor-intrinsic epithelial-mesenchymal transition and tumor-associated M2-like macrophage
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2023, 页码: 14
作者:
Pei, Jin-peng
;
Wang, Yue
;
Ma, Lan-ping
;
Wang, Xin
;
Liu, Liang
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2023/04/10
AXL
NSCLC
TNBC
M2-macrophage
antibody-drug conjugate
Five New Diarylbutyrolactones and Sesquilignans from Saussurea medusa and Their Inhibitory Effects on LPS-induced NO Production
期刊论文
OAI收割
PLANTA MEDICA, 2023, 页码: 11
作者:
Cao, Jing-Ya
;
Wang, Zhi-Yao
;
Stewart, Alan J. J.
;
Dong, Qi
;
Zhao, Ye
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2023/04/10
Saussurea medusa
Asteraceae
diarylbutyrolactone lignan
sesquilignan
anti-inflammatory activity
molecular docking
Megastigmane sesquiterpenoids from Saussurea medusa and their anti-inflammatory activities
期刊论文
OAI收割
NATURAL PRODUCT RESEARCH, 2022, 页码: 9
作者:
Cao, Jing-Ya
;
Dong, Qi
;
Wang, Zhi-Yao
;
Zhao, Ye
;
Ren, Yu
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2023/04/10
Saussurea medusa
megastigmane
sesquiterpenoid
anti-inflammatory activity
iNOS enzyme
Arylnaphthalide lignans from Saussurea medusa and their anti-inflammatory activities
期刊论文
OAI收割
ARABIAN JOURNAL OF CHEMISTRY, 2022, 卷号: 15, 期号: 10, 页码: 11
作者:
Cao, Jing-Ya
;
Dong, Qi
;
Wang, Zhi-Yao
;
Zhao, Ye
;
Ren, Yu
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2022/12/13
Saussurea medusa
Arylnaphthalide lignan
Anti-inflammatory activity
ECD calculation
Molecular docking
Rescue of maternal immune activation-induced behavioral abnormalities in adult mouse offspring by pathogen-activated maternal T-reg cells
期刊论文
OAI收割
NATURE NEUROSCIENCE, 2021, 页码: 33
作者:
Xu, Zhipeng
;
Zhang, Xiaoyun
;
Chang, Hao
;
Kong, Yue
;
Ni, Yangyue
  |  
收藏
  |  
浏览/下载:40/0
  |  
提交时间:2021/05/24
Two new neolignans and one new benzyl benzoate glycoside from Potentilla discolor
期刊论文
OAI收割
PHYTOCHEMISTRY LETTERS, 2020, 卷号: 39, 页码: 25-29
作者:
Wang, Wei
;
Ma, Xue-Jiao
;
Su, Yan-Fang
;
Gao, Zhi-Jing
;
Qin, Tao
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2021/05/24
Potentilla discolor
Chemical constituents
Neolignans
Benzyl benzoate glycoside
Leflunomide increased the renal exposure of acyclovir by inhibiting OAT1/3 and MRP2
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2020, 卷号: 41, 期号: 1, 页码: 129-137
作者:
Liao, Xiao-ying
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2020/07/01
leflunomide
teriflunomide
acyclovir
organic anion transporter
multidrug resistance associated protein (MRP) 2
drug-drug interaction
pharmacokinetics
Disulfide-Containing Detergents (DCDs) for the Structural Biology of Membrane Proteins
期刊论文
OAI收割
CHEMISTRY-A EUROPEAN JOURNAL, 2019, 页码: 7
作者:
Xue, Dongxiang
;
Xu, Tiandan
;
Wang, Huixia
;
Wu, Meng
;
Yuan, Ya
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2020/07/01
detergents
disulfides
membrane proteins
micelle size
NMR spectroscopy
Discovery of New Selective Butyrylcholinesterase (BChE) Inhibitors with Anti-A beta Aggregation Activity: Structure-Based Virtual Screening, Hit Optimization and Biological Evaluation
期刊论文
OAI收割
MOLECULES, 2019, 卷号: 24, 期号: 14, 页码: 21
作者:
Jiang, Cheng-Shi
;
Ge, Yong-Xi
;
Cheng, Zhi-Qiang
;
Wang, Yin-Yin
;
Tao, Hong-Rui
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2020/07/01
selective BChE inhibitor
virtual screening
structural optimization
molecular dynamics
anti-A beta aggregation