中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [19]
海洋研究所 [5]
心理研究所 [2]
上海生物化学与细胞生... [2]
上海营养与健康研究所 [2]
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期刊论文 [36]
会议论文 [1]
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2021 [2]
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Coronarin A modulated hepatic glycogen synthesis and gluconeogenesis via inhibiting mTORC1/S6K1 signaling and ameliorated glucose homeostasis of diabetic mice
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2022, 页码: 14
作者:
Huang, Su-Ling
;
Xie, Wei
;
Ye, Yang-Liang
  |  
收藏
  |  
浏览/下载:48/0
  |  
提交时间:2022/11/11
type 2 diabetes mellitus
coronarin A
glycogen synthesis
gluconeogenesis
mTORC1
IRS1
Structural basis of peptidomimetic agonism revealed by small-molecule GLP-1R agonists Boc5 and WB4-24
期刊论文
OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2022, 卷号: 119, 期号: 20, 页码: 10
作者:
Cong, Zhaotong
;
Zhou, Qingtong
;
Li, Yang
;
Chen, Li-Nan
;
Zhang, Zi-Chen
  |  
收藏
  |  
浏览/下载:41/0
  |  
提交时间:2022/09/30
glucagon-like peptide-1 receptor
type 2 diabetes mellitus
cryoelectron microscopy
peptidomimetic agonism
Discovery of 5-(3-bromo-2-(2,3-dibromo-4,5-dimethoxybenzyl)-4,5-dimethoxybenzylidene)thiazolidine-2,4-dione as a novel potent protein tyrosine phosphatase 1B inhibitor with antidiabetic properties
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2021, 卷号: 108, 页码: 13
作者:
Jiang, Bo
;
Luo, Jiao
;
Guo, Shuju
;
Wang, Lijun
  |  
收藏
  |  
浏览/下载:38/0
  |  
提交时间:2021/05/11
Type 2 diabetes mellitus
Protein tyrosine phosphatase 1B inhibitors
Thiazolidinedione
Insulin signaling
Anti-diabetic activities
Bitter Melon and Diabetes Mellitus
期刊论文
OAI收割
FOOD REVIEWS INTERNATIONAL, 2021
作者:
Gao,Ya
;
Li,Xian
;
Huang,Yanjie
;
Chen,Jianchao
;
Qiu,Minghua
  |  
收藏
  |  
浏览/下载:46/0
  |  
提交时间:2022/04/02
Bitter melon
diabetes mellitus
crude extracts
phyto-metabolites
hypoglycemic mechanism
MOMORDICA-CHARANTIA L.
11-BETA-HYDROXYSTEROID DEHYDROGENASE TYPE-1
ALPHA-GLUCOSIDASE INHIBITION
INSULIN-RESISTANCE
ANTIDIABETIC ACTIVITIES
GUT MICROBIOTA
STRUCTURAL-CHARACTERIZATION
PHENOLIC-COMPOUNDS
OXIDATIVE STRESS
PROTEIN-KINASE
Small molecule IVQ, as a prodrug of gluconeogenesis inhibitor QVO, efficiently ameliorates glucose homeostasis in type 2 diabetic mice
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2019, 卷号: 40, 期号: 9, 页码: 1193-1204
作者:
Zhou, Ting-ting
;
Zhao, Tong
;
Ma, Fei
;
Zhang, Yi-nan
;
Jiang, Jing
  |  
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2020/07/01
type 2 diabetes mellitus
hepatic gluconeogenesis
AMPK signaling pathway
(E)-3-(2-(quinoline-4-yl)vinyl)-1H-indol-6-ol (QVO)
4-[2-(1H-indol-3-yl)vinyl]quinoline (IVQ)
prodrug
D-ribose is elevated in T1DM patients and can be involved in the onset of encephalopathy
期刊论文
OAI收割
AGING-US, 2019, 卷号: 11, 期号: 14, 页码: 4943-4969
作者:
Yu, Lexiang
;
Chen, Yao
;
Xu, Yong
;
He, Tao
;
Wei, Yan
  |  
收藏
  |  
浏览/下载:68/0
  |  
提交时间:2019/10/25
D-ribose
benfotiamine (BTMP)
cognitive impairment
type 1 diabetic encephalopathy
type 1 diabetes mellitus (T1DM)
diabetic encephalopathy
Highly Selective Protein Tyrosine Phosphatase Inhibitor, 2,2 ',3,3 '-Tetrabromo-4,4 ',5,5 '-tetrahydroxydiphenylmethane, Ameliorates Type 2 Diabetes Mellitus in BKS db Mice
期刊论文
OAI收割
MOLECULAR PHARMACEUTICS, 2019, 卷号: 16, 期号: 5, 页码: 1839-1850
作者:
Li, Chao
;
Luo, Jiao
;
Guo, Shuju
;
Jia, Xiaoling
;
Guo, Chuanlong
  |  
收藏
  |  
浏览/下载:87/0
  |  
提交时间:2019/08/28
type 2 diabetes mellitus
protein tyrosine phosphatase 1B
insulin resistance
hypoglycemic activity
dyslipidemia
Synthesis and biological evaluation of novel potent FFA1 agonists containing 2,3-dihydrobenzo[b][1,4]dioxine
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2019, 卷号: 29, 期号: 6, 页码: 848-852
作者:
Kong, Deyu
;
Guo, Shimeng
;
Yang, Yushe
;
Guo, Bin
;
Xie, Xin
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2020/07/01
FFA1 agonist
2,3-Dihydrobenzo[b][1,4]dioxine
Insulin secretion
Type 2 diabetes mellitus
BMP10 suppresses hepatocellular carcinoma progression via PTPRS-STAT3 axis
期刊论文
OAI收割
ONCOGENE, 2019, 卷号: 38, 期号: 48, 页码: 7281-7293
作者:
Yuan, Yan-Mei
;
Ma, Ning
;
Zhang, Er-Bin
;
Chen, Tian-Wei
;
Jiang, Hao
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2020/12/09
Hematopoietic stem cell
Type 1 diabetes mellitus
Immune response
Th1 cell
Th17 cell
Regulartory T cell
Design and optimization of 2,3-dihydrobenzo[b][1,4]dioxine propanoic acids as novel GPR40 agonists with improved pharmacokinetic and safety profiles
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2018, 卷号: 26, 期号: 22, 页码: 5780-5791
作者:
Guo, Bin
;
Guo, Shimeng
;
Huang, Jing
;
Li, Jingya
;
Li, Jia
  |  
收藏
  |  
浏览/下载:62/0
  |  
提交时间:2019/01/08
GPR40 agonist
2,3-Dihydrobenzo[b][1,4]dioxine
Insulin secretion
Type 2 diabetes mellitus