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Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
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昆明植物研究所 [167]
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Discovery of novel SOS1 inhibitors using machine learning
期刊论文
OAI收割
RSC MEDICINAL CHEMISTRY, 2024, 卷号: 15, 期号: 4, 页码: 1392-1403
作者:
Duo, Lihui
;
Chen, Yi
;
Liu, Qiupei
;
Ma, Zhangyi
;
Farjudian, Amin
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2024/05/07
Development of Potent MALT1 Inhibitors Featuring a Novel "2-Thioxo-2,3-dihydrothiazolo[4,5-
d
]pyrimidin-7(6
H
)-one" Scaffold for the Treatment of B Cell Lymphoma
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 4, 页码: 2884-2906
作者:
Liang, Xuewu
;
Yu, Haolan
;
Liang, Renwen
;
Feng, Zhuanghui
;
Saidahmatov, Abdusaid
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2024/04/09
Cloning and functional characterization of the oxidative squalene cyclase gene in the deep-sea holothurian Chiridota sp.
期刊论文
OAI收割
GENE, 2024, 卷号: 894, 页码: 9
作者:
Huang, Yanan
;
Liu, Helu
;
Zhou, Yang
;
Lu, Zaiqing
;
Pu, Yujin
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2024/01/08
Deep-sea
Holothurian
Chiridota sp
Sea cucumber triterpenes
GC -MS
Discovery of a 1,6-naphthyridin-4-one-based AXL inhibitor with improved pharmacokinetics and enhanced in vivo antitumor efficacy
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 265, 页码: 17
作者:
Lan, Yaohan
;
Peng, Xia
;
Ji, Yinchun
;
Su, Yi
;
Duan, Wenhu
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2024/02/27
AXL inhibitor
In vivo antitumor efficacy
6-Naphthyridin-4-one derivatives
Scaffold hopping
Structure-based drug design
Structure-based identification of new orally bioavailable BRD9-PROTACs for treating acute myelocytic leukemia
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 262, 页码: 18
作者:
Zhang, Jingyu
;
Duan, Haiting
;
Gui, Renzhao
;
Wu, Mingfei
;
Shen, Liteng
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2023/12/19
Acute myeloid leukemia
Bromodomain-containing protein 9
Proteolysis-targeting chimera
Orally bioavailable
Docking
The
Ginkgo biloba
L. in China: Current Distribution and Possible Future Habitat
期刊论文
OAI收割
FORESTS, 2023, 卷号: 14, 期号: 12, 页码: 18
作者:
Zhang, Ying
;
Zhang, Jinbing
;
Tian, Li
;
Huang, Yaohui
;
Shao, Changliang
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2024/01/22
Ginkgo biloba L.
climate change
MaxEnt
climate change scenario
China
The Ginkgo biloba L. in China: Current Distribution and Possible Future Habitat
期刊论文
OAI收割
FORESTS, 2023, 卷号: 14, 期号: 12, 页码: 2284
作者:
Zhang, Ying
;
Zhang, Jinbing
;
Tian, Li
;
Huang, Yaohui
;
Shao, Changliang
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2024/01/26
Ginkgo biloba L.
climate change
MaxEnt
climate change scenario
China
Design, Synthesis, and Pharmacological Evaluation of Isoindoline Analogues as New HPK1 Inhibitors
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 23, 页码: 16201-16221
作者:
Xie, Chenghu
;
Liu, Bo
;
Song, Zilan
;
Yang, Ye
;
Dai, Mengdi
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2024/02/27
Discovery, structural optimization, and anti-tumor bioactivity evaluations of betulinic acid derivatives as a new type of ROR & gamma; antagonists
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 257, 页码: 15
作者:
Mei, Lianghe
;
Xu, Lansong
;
Wu, Sanan
;
Wang, Yafang
;
Xu, Chao
  |  
收藏
  |  
浏览/下载:40/0
  |  
提交时间:2023/10/17
Betulinic acid
ROR & gamma
Target identification
Rationale structure optimization
Anti-tumor effects
antagonists
Discovery and Mechanism Study of SARS-CoV-2 3C-like Protease Inhibitors with a New Reactive Group
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 页码: 18
作者:
Ren, Pengxuan
;
Li, Hui
;
Nie, Tianqing
;
Jian, Xiaoqin
;
Yu, Changyue
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2023/10/17