中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共138条,第1-10条 帮助

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Identification of Dihydrobenzofuran Neolignans as Novel PDE4 Inhibitors and Evaluation of Antiatopic Dermatitis Efficacy in DNCB-Induced Mice Model 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 6, 页码: 4855-4869
作者:  
Gu, Chenming;  Liu, Jiayuan;  Qian, Fei;  Yu, Wenchao;  Huang, Doudou
  |  收藏  |  浏览/下载:1/0  |  提交时间:2024/05/07
Ecto-nucleotide pyrophosphatase/phosphodiesterase 1 inhibitors: Research progress and prospects 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 267, 页码: 13
作者:  
Guan, Dezhong;  Fang, Lincheng;  Feng, Mingshun;  Guo, Shi;  Xie, Lingfeng
  |  收藏  |  浏览/下载:1/0  |  提交时间:2024/05/07
Ent-labdane-type diterpene glycosides obtained from Rubus chingii Hu and their inhibitory effects on PDE5A activity 期刊论文  OAI收割
FITOTERAPIA, 2024, 卷号: 173, 页码: 14
作者:  
Yu, Jun-dong;  Wang, Jing-Yi;  Liu, Jia-yuan;  Xu, Ye-chun;  Zhang, Xue
  |  收藏  |  浏览/下载:12/0  |  提交时间:2024/02/27
Discovery of Pyrido[2,3-d]pyrimidin-7-one Derivatives as Highly Potent and Efficacious Ectonucleotide Pyrophosphatase/Phosphodiesterase 1 (ENPP1) Inhibitors for Cancer Treatment 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 5, 页码: 3986-4006
作者:  
Sun, Yaoliang;  Chen, Manman;  Han, Yuyan;  Li, Weiqiang;  Ma, Xiaoyu
  |  收藏  |  浏览/下载:1/0  |  提交时间:2024/05/07
Drug repurposing and structure-based discovery of new PDE4 and PDE5 inhibitors 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 262, 页码: 14
作者:  
Liu, Jiayuan;  Zhang, Xianglei;  Chen, Guofeng;  Shao, Qiang;  Zou, Yi
  |  收藏  |  浏览/下载:22/0  |  提交时间:2024/01/16
Phylogenetic Analysis and Characterization of Diguanylate Cyclase and Phosphodiesterase in Planktonic Filamentous Cyanobacterium Arthrospira sp. 期刊论文  OAI收割
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 2023, 卷号: 24, 期号: 20, 页码: 11
作者:  
Wang, Kang;  Li, Wenjun;  Cui, Hongli;  Qin, Song
  |  收藏  |  浏览/下载:20/0  |  提交时间:2024/01/26
Bioactive compounds from Huashi Baidu decoction possess both antiviral and anti-inflammatory effects against COVID-19 期刊论文  OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2023, 卷号: 120, 期号: 18, 页码: 11
作者:  
Xu, Haiyu;  Li, Shufen;  Liu, Jiayuan;  Cheng, Jinlong;  Kang, Liping
  |  收藏  |  浏览/下载:21/0  |  提交时间:2023/10/17
Pharmacokinetics,mass balance,and metabolism of 14C TPN171,a novel PDE5 inhibitor,in humans for the treatment of pulmonary arterial hypertension 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2023, 卷号: 44, 期号: 1, 页码: 221
作者:  
He Yifei;  Liu Yin;  Yu Jinghua;  Cheng Huan;  Odilov Abdullajon
  |  收藏  |  浏览/下载:15/0  |  提交时间:2023/05/22
Magnetic multi-enzyme cascade combined with liquid chromatography tandem mass spectrometry for fast DNA digestion and quantitative analysis of 5-hydroxymethylcytosine in genome of human bladder cancer T24 cells induced by tetrachlorobenzoquinone 期刊论文  OAI收割
JOURNAL OF CHROMATOGRAPHY A, 2022, 卷号: 1676, 期号: 0, 页码: 463279
作者:  
Fang, Tianjiao;  Tang, Chao;  Yin, Junfa;  Wang, Hailin
  |  收藏  |  浏览/下载:15/0  |  提交时间:2022/11/08
TPN171H alleviates pulmonary hypertension via inhibiting inflammation in hypoxia and monocrotaline-induced rats 期刊论文  OAI收割
VASCULAR PHARMACOLOGY, 2022, 卷号: 145, 页码: 11
作者:  
Zhao, Congke;  Hu, Liqing;  He, Xiangrong;  Li, Lijun;  Yin, Minghui
  |  收藏  |  浏览/下载:33/0  |  提交时间:2022/08/16