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上海药物研究所 [58]
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Ent-labdane-type diterpene glycosides obtained from
Rubus
chingii
Hu and their inhibitory effects on PDE5A activity
期刊论文
OAI收割
FITOTERAPIA, 2024, 卷号: 173, 页码: 14
作者:
Yu, Jun-dong
;
Wang, Jing-Yi
;
Liu, Jia-yuan
;
Xu, Ye-chun
;
Zhang, Xue
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2024/02/27
diterpene glycosides
Rubus Chingii Hu
PDE5A inhibitory activity
ent-labdane
Drug repurposing and structure-based discovery of new PDE4 and PDE5 inhibitors
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 262, 页码: 14
作者:
Liu, Jiayuan
;
Zhang, Xianglei
;
Chen, Guofeng
;
Shao, Qiang
;
Zou, Yi
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2024/01/16
Phosphodiesterase-4 (PDE4)
PDE5
Inhibitor
Drug repurposing
Crystal structure
Structure -guided optimization
Phylogenetic Analysis and Characterization of Diguanylate Cyclase and Phosphodiesterase in Planktonic Filamentous Cyanobacterium
Arthrospira
sp.
期刊论文
OAI收割
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 2023, 卷号: 24, 期号: 20, 页码: 11
作者:
Wang, Kang
;
Li, Wenjun
;
Cui, Hongli
;
Qin, Song
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2024/01/26
c-di-GMP
Arthrospira
diguanylate cyclase
phosphodiesterase
riboswitch
Bioactive compounds from Huashi Baidu decoction possess both antiviral and anti-inflammatory effects against COVID-19
期刊论文
OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2023, 卷号: 120, 期号: 18, 页码: 11
作者:
Xu, Haiyu
;
Li, Shufen
;
Liu, Jiayuan
;
Cheng, Jinlong
;
Kang, Liping
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2023/10/17
COVID-19
traditional Chinese medicine
TCMT-NDRD
antivirus
anti-inflammation
Pharmacokinetics,mass balance,and metabolism of 14C TPN171,a novel PDE5 inhibitor,in humans for the treatment of pulmonary arterial hypertension
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2023, 卷号: 44, 期号: 1, 页码: 221
作者:
He Yifei
;
Liu Yin
;
Yu Jinghua
;
Cheng Huan
;
Odilov Abdullajon
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2023/05/22
TPN171
14CTPN171
PDE5 inhibitor
pulmonary arterial hypertension
healthy volunteers
pharmacokinetics
metabolite identification
mass balance
Magnetic multi-enzyme cascade combined with liquid chromatography tandem mass spectrometry for fast DNA digestion and quantitative analysis of 5-hydroxymethylcytosine in genome of human bladder cancer T24 cells induced by tetrachlorobenzoquinone
期刊论文
OAI收割
JOURNAL OF CHROMATOGRAPHY A, 2022, 卷号: 1676, 期号: 0, 页码: 463279
作者:
Fang, Tianjiao
;
Tang, Chao
;
Yin, Junfa
;
Wang, Hailin
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2022/11/08
DISINFECTION BY-PRODUCTS
METAL-ORGANIC FRAMEWORKS
BROMO-BENZOQUINONES
ADDUCTS
HALOBENZOQUINONES
ENZYMES
TPN171H alleviates pulmonary hypertension via inhibiting inflammation in hypoxia and monocrotaline-induced rats
期刊论文
OAI收割
VASCULAR PHARMACOLOGY, 2022, 卷号: 145, 页码: 11
作者:
Zhao, Congke
;
Hu, Liqing
;
He, Xiangrong
;
Li, Lijun
;
Yin, Minghui
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2022/08/16
Pulmonary hypertension
Hypoxia
Monocrotaline
Anti-inflammatory effects
NLRP3 inflammasome
Pulmonary artery endothelial cells
Pharmacokinetics, mass balance, and metabolism of [C-14]TPN171, a novel PDE5 inhibitor, in humans for the treatment of pulmonary arterial hypertension
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2022, 页码: 13
作者:
He, Yi-fei
;
Liu, Yin
;
Yu, Jing-hua
;
Cheng, Huan
;
Odilov, Abdullajon
  |  
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2022/08/16
TPN171
[C-14]TPN171
PDE5 inhibitor
pulmonary arterial hypertension
healthy volunteers
pharmacokinetics
metabolite identification
mass balance
Absorption, distribution, metabolism, and excretion of [C-14]TPN729 after oral administration to rats
期刊论文
OAI收割
XENOBIOTICA, 2022, 页码: 12
作者:
Cheng, Huan
;
Yu, Jinghua
;
Yang, Chen
;
Zhang, Ning
;
Fan, Zhen
  |  
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2022/06/15
TPN729
[C-14]TPN729
mass balance
tissue distribution
metabolism
Targeting PDE4 as a promising therapeutic strategy in chronic ulcerative colitis through modulating mucosal homeostasis
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2022, 卷号: 12, 期号: 1, 页码: 228-245
作者:
Li, Heng
;
Zhang, Yao
;
Liu, Moting
;
Fan, Chen
;
Feng, Chunlan
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2022/06/15
Ulcerative colitis
Mucosal homeostasis
Gut microbiota
Epithelial barrier
PDE4